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BML-277
A selective DNA damage control kinase inhibitor
GDC-0575 (ARRY-575, RG7741)
A Chk1 inhibitor
GDC-0575 dihydrochloride (ARRY-575 dihydrochloride)
LY2606368
CHK1-IN-3
CHK1-IN-3 是一種檢測點(diǎn)激酶 (CHK1) 抑制劑,IC50 值為 0.4 nM。
Debromohymenialdisine
An inhibitor of Chk1 and Chk2
CCT241533 hydrochloride
A selective Chk2 inhibitor
CCT245737
A potent Chk1 inhibitor
LY2603618
CCT241533
PD 407824
An inhibitor of Chk1 and WEE1
ML367
ML367 is a potent, micromolar inhibitor of ATPase family AAA domain-containing protein 5 (ATAD5) stabilization. ML367 blocks DNA repair pathways and general DNA damage responses including RPA32-phosphorylation and CHK1-phosphorylation in response to UV ir
CHK-IN-1
CHK-IN-1是一種CHK1和CHK2的抑制劑,具有抗增殖作用。
Chk2 Inhibitor
A Chk2 inhibitor
Prexasertib Mesylate Hydrate
Prexasertib Mesylate Hydrate (LY2606368 Mesylate Hydrate) 是一種有效、選擇性、 ATP 競爭性的 CHK1 和 CHK2 抑制劑,對 CHK1 的 Ki 值為 0.9 nM,IC50 值 <1 nM,對 CHK2 的 IC50 值為 8 nM。Prexasertib Mesylate Hydrate 抑制 HT-29 細(xì)胞 CHK1 (S296) 和 CHK2 (S516) 的自身磷酸化。Prexasertib Mesylate Hydrate 具
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