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Trilaciclib (G1T28)
Trilaciclib (G1T28, G1T28-1) is a highly potent, selective and reversible cyclin-dependent kinase 4 and 6 (CDK4/6) inhibitor. Trilaciclib inhibits CDK4/cyclin D1 and CDK6/cyclin D3 with IC50 of 1 nM and 4 nM, respectively.
PHA-793887
A CDK inhibitor
CDK4/6-IN-2
CDK4/6-IN-2 是一種有效的 CDK4 和 CDK6 抑制劑,IC50 分別為 2.7 和 16 nM,詳細信息請參考專利文獻 US20180000819A1 中 的化合物 1。
Ribociclib succinate hydrate
Ribociclib (LEE011) succinate (Kisqali) is a highly specific dual inhibitor of CDK4 and CDK6 with IC50 of 10 nM and 39 nM, respectively.
Ro 3306
An inhibitor of Cdk1
PHA-767491
A potent Cdc7 kinase inhibitor
PF-06873600
An inhibitor of Cdk2, Cdk4, and Cdk6
LDC4297
A CDK7 inhibitor
CDK4 inhibitor
An antiproliferative cyclin D1/Cdk4 inhibitor
Cucurbitacin D
A triterpenoid with diverse biological activities
FMF-04-159-2
FMF-04-159-2 是一種有效的共價 CDK14 抑制劑。FMF-04-159-2 抑制 CDK14 和 CDK2,在 NanoBRET 試驗中 IC50 分別為 39.6 nM 和 256 nM。
Senexin B
An inhibitor of Cdk8 and Cdk19
Indirubin-5-sulfonate
Indirubin-5-sulfonate 是周期蛋白依賴性激酶(CDK) 的抑制劑,對CDK1/cyclin B、CDK2/cyclin A、CDK2/cyclin E、CDK4/cyclin D1 和CDK5/p35 的IC50 值分別為55 nM、35 nM、150 nM、300 nM 和 65 nM。Indirubin-5-sulfonate 同樣能抑制GSK-3β 的活性。
(-)-BAY-1251152
A racemic mixture of (+)-BAY-1251152 and (–)-BAY-1251152
PHA-767491 hydrochloride
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